Fluorescent M3 antagonist [pirenzepine] (AC128)
Cat.#: ASSD-128
Inquiry
Specifications
Description |
Fluorescent M3 muscarinic receptor antagonist (apparent KD values are 7.97, 6.29 and 6.24 for M3, M5 and M1 receptors respectively). Antagonizes the activity of carbachol, a muscarinic receptor agonist. Displays no intrinsic activity. |
Synonyms |
M3-633-AN |
Size |
50 μg |
Applications |
For imaging at the M3 receptor use solutions up to 100 nM. |
Molecule Weight |
1014 |
Purity |
>97% |
Solubility |
Soluble in DMSO |
Excitation |
633 nm |
Emission |
650 nm |
Storage |
Store at -20° C |
Shipping |
Shipped at 4°C |
Important |
We strongly recommend storing this product away from light and briefly sonicating the sample when using to ensure it is fully dissolved and the solution is homogeneous. However, we do not recommend using the product after subjecting it to repetitive freeze-thaw cycles. |
Related Products
All of our products
are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.