Fluorescent adenosine A3 antagonist [XAC] (AC121)
Cat.#: ASSD-121
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Specifications
Description |
Fluorescent A3 adenosine receptor antagonist. Displays selectivity for A3 over A2A and A1 (apparent KD values are 8.10, 6.74 and 6.57 respectively). Antagonizes the activity of NECA, an adenosine receptor agonist. Exhibits no intrinsic agonist activity. A fluorescent Xanthine Amine Congener (XAC) analog. |
Synonyms |
Fluorescent Adenosine A3 receptor Antagonist (A3-633-AN), A3-633-AN |
Size |
500 μg |
Applications |
For ligand binding; fluorescence imaging; high content analysis; kinetic analysis; cell sorting at adenosine A1 / A2A / A3 receptors use solutions up to 100 nM. |
Molecule Weight |
1144 |
Purity |
>95% |
Solubility |
Soluble in DMSO |
Form |
Purple solid |
Excitation |
633 nm |
Emission |
650 nm |
Storage |
Store at -20° C(protect from light) |
Shipping |
Shipped at 4°C |
Important |
We recommend briefly sonicating the sample when using to ensure it is fully dissolved and the solution is homogeneous. However, we do not recommend using the product after subjecting it to repetitive freeze-thaw cycles. |
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are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.