Related Diseases
Depression
Description
TASP0233278 is a potent and orally active V1B receptor antagonist with antidepressant and anxiolytic activities in rodents.
Chemical Formula
C30H31ClFN3O7S
Molecular Weight
632.1004
Elemental Analysis
C, 57.01; H, 4.94; Cl, 5.61; F, 3.01; N, 6.65; O, 17.72; S, 5.07
Synonym
TASP0233278; TASP 0233278; TASP-0233278;
IUPAC/Chemical Name
(2S,4R)-1-((R)-5-chloro-1-((2,4-dimethoxyphenyl)sulfonyl)-3-(2-methoxyphenyl)-2-oxoindolin-3-yl)-4-fluoro-N,N-dimethylpyrrolidine-2-carboxamide
InChi Key
DKGOINZYRASALR-WEWKHQNJSA-N
InChi Code
InChI=1S/C30H31ClFN3O7S/c1-33(2)28(36)24-15-19(32)17-34(24)30(21-8-6-7-9-25(21)41-4)22-14-18(31)10-12-23(22)35(29(30)37)43(38,39)27-13-11-20(40-3)16-26(27)42-5/h6-14,16,19,24H,15,17H2,1-5H3/t19-,24+,30+/m1/s1
SMILES Code
O=C(N1S(=O)(C2=CC=C(OC)C=C2OC)=O)[C@](N3C[C@H](F)C[C@H]3C(N(C)C)=O)(C4=CC=CC=C4OC)C5=C1C=CC(Cl)=C5
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
To be determined
Shelf Life
>2 years if stored properly
Drug Formulation
To be determined
Stock Solution Storage
0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).
HS Tariff Code
2934.99.9001