Related Diseases
Depression
Product Name
Tampramine fumarate
Description
Tampramine (AHR-9,377) is a tricyclic antidepressant (TCA) which was developed in the 1980s but was never marketed. Despite being a TCA, it acts as a selective norepinephrine reuptake inhibitor and has negligible affinity for adrenergic, histaminergic, and muscarinic receptors.
Chemical Formula
C27H28N4O4
Elemental Analysis
C, 68.63; H, 5.97; N, 11.86; O, 13.54
Synonym
Tampramine fumarate; AHR 9377; AHR-9377; AHR9377
IUPAC/Chemical Name
11H-Pyrido(2,3-b)(1,4)benzodiazepine-11-propanamine, N,N-dimethyl-6-phenyl-, (E)-2-butenedioate (1:1)
InChi Key
USQAILMOWHOBTK-WLHGVMLRSA-N
InChi Code
InChI=1S/C23H24N4.C4H4O4/c1-26(2)16-9-17-27-21-14-7-6-12-19(21)22(18-10-4-3-5-11-18)25-20-13-8-15-24-23(20)27;5-3(6)1-2-4(7)8/h3-8,10-15H,9,16-17H2,1-2H3;1-2H,(H,5,6)(H,7,8)/b;2-1+
SMILES Code
CN(C)CCCN1C2=NC=CC=C2N=C(C3=CC=CC=C3)C4=CC=CC=C41.O=C(O)/C=C/C(O)=O
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).
HS Tariff Code
2934.99.9001