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Sunepitron HCl

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Specification

Cat. No.

SMD390

Related Diseases

Anxiety

Product Name

Sunepitron HCl

Size

5.0mg; 25.0mg

Price

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Availability

2 Weeks

Description

Sunepitron, also known as CP-93,393 or CP-93,393-1 (HCl), is a combined 5-HT1A receptor agonist and α2-adrenergic receptor antagonist. It was previously under development by Pfizer for the treatment of depression and anxiety. It made it to phase III clinical trials before being discontinued.

CAS Number

148408-65-5 (HCl)

Chemical Formula

C17H24ClN5O2

Molecular Weight

365.862

Elemental Analysis

C, 55.81; H, 6.61; Cl, 9.69; N, 19.14; O, 8.75

Synonym

CP-93,393; CP 93,393; CP93,393; CP-93393; CP 93393; CP93393; CP-93,393-1; Sunepitron. Sunepitron HCl.

IUPAC/Chemical Name

1-(((7S,9aS)-2-(pyrimidin-2-yl)octahydro-2H-pyrido[1,2-a]pyrazin-7-yl)methyl)pyrrolidine-2,5-dione hydrochloride

InChi Key

HWGPYTRJVVMHGT-IODNYQNNSA-N

InChi Code

InChI=1S/C17H23N5O2.ClH/c23-15-4-5-16(24)22(15)11-13-2-3-14-12-21(9-8-20(14)10-13)17-18-6-1-7-19-17;/h1,6-7,13-14H,2-5,8-12H2;1H/t13-,14-;/m0./s1

SMILES Code

O=C(N1C[C@H]2CC[C@@]3([H])CN(C4=NC=CC=N4)CCN3C2)CCC1=O.[H]Cl

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.