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Sunepitron Free Base

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Specification

Cat. No.

SMD377

Related Diseases

Anxiety

Product Name

Sunepitron Free Base

Size

Customizable

Price

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Description

Sunepitron Free Base is a combined 5-HT1A receptor agonist and α₂-adrenergic receptor antagonist. It was previously under development by Pfizer for the treatment of depression and anxiety. It made it to phase III clinical trials before being discontinued.

CAS Number

131831-03-3 (free base)

Chemical Formula

C17H23N5O2

Exact Mass

329.1852

Molecular Weight

329.4

Elemental Analysis

C, 61.99; H, 7.04; N, 21.26; O, 9.71

Synonym

Sunepitron Free Base; CP93,393; CP 93,393; CP-93,393

IUPAC/Chemical Name

2,5-Pyrrolidinedione, 1-(((7S,9aS)-octahydro-2-(2-pyrimidinyl)-2H-pyrido(1,2-a)pyrazin-7-yl)methyl)-

InChi Key

UXWBIYCPUVWKHP-KBPBESRZSA-N

InChi Code

InChI=1S/C17H23N5O2/c23-15-4-5-16(24)22(15)11-13-2-3-14-12-21(9-8-20(14)10-13)17-18-6-1-7-19-17/h1,6-7,13-14H,2-5,8-12H2/t13-,14-/m0/s1

SMILES Code

O=C(CC1)N(C[C@H]2CC[C@@]3([H])CN(C4=NC=CC=N4)CCN3C2)C1=O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.