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SR-12062

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Specification

Cat. No.

SMD1709

Related Diseases

Schizophrenia

Product Name

SR-12062

Size

Customizable

Price

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Description

SR-12062 is a full agonists of the neurotensin receptor 1 (NTSR1). SR-12062 have an EC50 of 2 μM at NTSR1 with full agonist behaviour (Emax=100%), showing a higher efficacy and ∼90-fold potency improvement compared to parent compound 1 (EC50=178 μM; Emax=17%).

CAS Number

1623019-77-1

Chemical Formula

C25H25N3O3

Exact Mass

415.1896

Molecular Weight

415.493

Elemental Analysis

C, 72.27; H, 6.07; N, 10.11; O, 11.55

Synonym

SR-12062; SR 12062; SR12062;

IUPAC/Chemical Name

(2-(5-(quinolin-3-yl)-1H-indol-1-yl)acetyl)-L-leucine

InChi Key

FPIZUBHJQMKCPU-QFIPXVFZSA-N

InChi Code

InChI=1S/C25H25N3O3/c1-16(2)11-22(25(30)31)27-24(29)15-28-10-9-19-12-17(7-8-23(19)28)20-13-18-5-3-4-6-21(18)26-14-20/h3-10,12-14,16,22H,11,15H2,1-2H3,(H,27,29)(H,30,31)/t22-/m0/s1

SMILES Code

O=C(N[C@@H](CC(C)C)C(O)=O)CN1C=CC2=C1C=CC(C3=CC4=CC=CC=C4N=C3)=C2

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>3 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.