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Pipofezine HCl

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Specification

Cat. No.

SMD1128

Related Diseases

Depression

Product Name

Pipofezine HCl

Size

Customizable

Price

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Description

Pipofezine, also known as Azafen or Azaphen, is a tricyclic antidepressant (TCA) approved in Russia for the treatment of depression. It was introduced in the late 1960s and is still used today. Pipofezine has been shown to act as a potent inhibitor of the reuptake of serotonin. In addition to its antidepressant action, pipofezine has sedative effects as well, suggesting antihistamine activity. Other properties such as anticholinergic or antiadrenergic actions are less clear but are likely.

CAS Number

24853-80-3 (HCl)

Chemical Formula

C16H20ClN5O

Molecular Weight

333.82

Elemental Analysis

C, 57.57; H, 6.04; Cl, 10.62; N, 20.98; O, 4.79

Synonym

Azaphen HCl; Azafen; Pipofezine; Pipofezine HCl

IUPAC/Chemical Name

5-methyl-3-(4-methylpiperazin-1-yl)pyridazino[3,4-b][1,4]benzoxazine hydrochloride.

InChi Key

JVONTAXIALFQJM-UHFFFAOYSA-N

InChi Code

InChI=1S/C16H19N5O.ClH/c1-19-7-9-21(10-8-19)15-11-13-16(18-17-15)22-14-6-4-3-5-12(14)20(13)2;/h3-6,11H,7-10H2,1-2H3;1H

SMILES Code

CN1CCN(C2=NN=C3OC4=CC=CC=C4N(C)C3=C2)CC1.[H]Cl

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO, not in water

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.