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Pipequaline HCl

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Specification

Cat. No.

SMD355

Related Diseases

Anxiety

Product Name

Pipequaline HCl

Size

100.0mg; 200.0mg; 500.0mg; 1.0g; 2.0g; 5.0g

Price

Inquiry

Availability

2 Weeks

Description

Pipequaline, also known as PK-8165, is an anxiolytic drug that was never marketed. It possesses a novel chemical structure that is not closely related to other drugs of this type. The drug has a similar pharmacological profile to the benzodiazepine family of drugs, but with mainly anxiolytic properties and very little sedative, amnestic or anticonvulsant effects, and so is classified as a nonbenzodiazepine anxiolytic. Pipequaline acts as a non-selective GABAA receptor partial agonist. While its profile of anxiolytic effects without sedation would appear to have potential medical applications, pipequaline has never been developed for medical use and is currently only used in scientific research.

CAS Number

80221-58-5 (HCl)

Chemical Formula

C22H25ClN2

Exact Mass

316.1939

Molecular Weight

352.906

Elemental Analysis

C, 74.88; H, 7.14; Cl, 10.05; N, 7.94

Synonym

Pipequaline; PK 8165; PK-8165; PK8165; Pipequaline HCl; Pipequaline hydrochloride

IUPAC/Chemical Name

2-Phenyl-4-(2-(4-piperidinyl)ethyl)quinoline monohydrochloride

InChi Key

JWEMPGHGMSUJIS-UHFFFAOYSA-N

InChi Code

InChI=1S/C22H24N2.ClH/c1-2-6-18(7-3-1)22-16-19(11-10-17-12-14-23-15-13-17)20-8-4-5-9-21(20)24-22;/h1-9,16-17,23H,10-15H2;1H

SMILES Code

[H]Cl.C1(C2=CC=CC=C2)=NC3=CC=CC=C3C(CCC4CCNCC4)=C1

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.