Related Diseases
Depression
Size
50.0mg; 100.0mg; 200.0mg; 500.0mg; 1.0g; 2.0g
Description
NS-5806 is a KV4.3 channel activator. It acts by mediating the transient outward K+ current (Ito) and increasing IKv4.3 peak current amplitude in CHO-K1 cells expressing KV4.3 and KChIP2.
Chemical Formula
C16H8Br2F6N6O
Molecular Weight
574.0794
Elemental Analysis
C, 33.48; H, 1.40; Br, 27.84; F, 19.86; N, 14.64; O, 2.79
Synonym
NS-5806; NS 5806; NS5806;
IUPAC/Chemical Name
1-[3,5-Bis(trifluoromethyl)phenyl]-3-[2,4-dibromo-6-(2H-tetrazol-5-yl)phenyl]urea
InChi Key
UZWJWROOLOOCPQ-UHFFFAOYSA-N
InChi Code
InChI=1S/C16H8Br2F6N6O/c17-8-4-10(13-27-29-30-28-13)12(11(18)5-8)26-14(31)25-9-2-6(15(19,20)21)1-7(3-9)16(22,23)24/h1-5H,(H2,25,26,31)(H,27,28,29,30)
SMILES Code
O=C(NC1=C(C2=NNN=N2)C=C(Br)C=C1Br)NC3=CC(C(F)(F)F)=CC(C(F)(F)F)=C3
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).
HS Tariff Code
2934.99.03.00