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MRS2365 sodium

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Specification

Cat. No.

SMD1026

Related Diseases

Depression

Product Name

MRS2365 sodium

Size

1.0mg

Price

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Availability

2 Weeks

Description

MRS2365 is a highly potent and selective P2Y1 receptor agonist (EC50 = 0.4 nM). MRS2365 displays no activity at P2Y12 receptors and only very low agonist activity at P2Y13 receptors (at concentrations up to 1 μM). MRS2365 increases the upregulation of NTPDase1 by ATPγS.

CAS Number

MRS2365 sodium

Chemical Formula

C13H16N5Na3O9P2S

Exact Mass

548.9837

Molecular Weight

549.27

Elemental Analysis

C, 28.43; H, 2.94; N, 12.75; Na, 12.56; O, 26.21; P, 11.28; S, 5.84

Synonym

MRS2365; MRS 2365; MRS-2365; (N)-methanocarba-2MeSADP;

IUPAC/Chemical Name

[(1R,2R,3S,5S)-4-[6-amino-2-(methylsulfanyl)-9H-purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexan-1-yl]methyl sodium {[bis(sodiooxy)phosphoryl]oxy}phosphonate

InChi Key

ZYPJOXVKTCEBCA-PVMCGCOJSA-K

InChi Code

InChI=1S/C13H19N5O9P2S.3Na/c1-30-12-16-10(14)6-11(17-12)18(4-15-6)7-5-2-13(5,9(20)8(7)19)3-26-29(24,25)27-28(21,22)23;;;/h4-5,7-9,19-20H,2-3H2,1H3,(H,24,25)(H2,14,16,17)(H2,21,22,23);;;/q;3*+1/p-3/t5-,7?,8+,9+,13+;;;/m1.../s1

SMILES Code

O=P(OP(OC[C@]12[C@@H](O)[C@@H](O)C(N3C=NC4=C(N)N=C(SC)N=C34)[C@@]1([H])C2)([O-])=O)(O[Na])O[Na].[Na+]

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.