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MPX-007

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Specification

Cat. No.

SMD522

Related Diseases

Autism

Related Diseases

Schizophrenia

Product Name

MPX-007

Size

Customizable

Price

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Description

MPX-007 is a potent NMDA inhibitor. MPX-007 inhibit GluN2A-containing NMDA receptors expressed in HEK cells with IC50s of 27 nM. MPX-007 offer highly selective pharmacological tools to probe GluN2A physiology and involvement in neuropsychiatric and developmental disorders.

CAS Number

1688685-29-1

Chemical Formula

C18H17F2N5O3S2

Exact Mass

453.0741

Molecular Weight

453.4828

Elemental Analysis

C, 47.68; H, 3.78; F, 8.38; N, 15.44; O, 10.58; S, 14.14

Synonym

MPX-007; MPX 007; MPX007.

IUPAC/Chemical Name

5-(((3,4-difluorophenyl)sulfonamido)methyl)-6-methyl-N-((2-methylthiazol-5-yl)methyl)pyrazine-2-carboxamide

InChi Key

GZXSPNTWOSSNMG-UHFFFAOYSA-N

InChi Code

InChI=1S/C18H17F2N5O3S2/c1-10-16(9-24-30(27,28)13-3-4-14(19)15(20)5-13)22-8-17(25-10)18(26)23-7-12-6-21-11(2)29-12/h3-6,8,24H,7,9H2,1-2H3,(H,23,26)

SMILES Code

O=C(C1=NC(C)=C(CNS(=O)(C2=CC=C(F)C(F)=C2)=O)N=C1)NCC3=CN=C(C)S3

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.