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MGS0274 besylate

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Specification

Cat. No.

SMD1577

Related Diseases

Schizophrenia

Product Name

MGS0274 besylate

Size

Customizable

Price

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Description

MGS0274 besylate is a prodrug of a potent group II metabotropic glutamate receptor agonist MGS0008 for the treatment of schizophrenia.

CAS Number

1501974-74-8 (besylate)

Chemical Formula

C27H38FNO10S

Exact Mass

587.22

Molecular Weight

587.6564

Elemental Analysis

C, 55.18; H, 6.52; F, 3.23; N, 2.38; O, 27.23; S, 5.46

Synonym

MGS0274 besylate; MGS 0274 besylate; MGS-0274 besylate; TS-134; TS134; TS 134;

IUPAC/Chemical Name

(1S,2S,3S,5R,6S)-2-amino-3-fluoro-6-(((S)-1-(((((1R,2S,5R)-2-isopropyl-5-methylcyclohexyl)oxy)carbonyl)oxy)ethoxy)carbonyl)bicyclo[3.1.0]hexane-2-carboxylic acid compound with benzenesulfonic acid (1:1)

InChi Key

KBBPYUNXSHDAMX-UDOTWNLBSA-N

InChi Code

InChI=1S/C21H32FNO7.C6H6O3S/c1-9(2)12-6-5-10(3)7-14(12)30-20(27)29-11(4)28-18(24)16-13-8-15(22)21(23,17(13)16)19(25)26;7-10(8,9)6-4-2-1-3-5-6/h9-17H,5-8,23H2,1-4H3,(H,25,26);1-5H,(H,7,8,9)/t10-,11+,12+,13+,14-,15+,16+,17+,21+;/m1./s1

SMILES Code

O=S(C1=CC=CC=C1)(O)=O.O=C([C@H]2[C@H]3[C@@H]2[C@](N)(C(O)=O)[C@@H](F)C3)O[C@H](C)OC(O[C@@H]4C[C@H](C)CC[C@H]4C(C)C)=O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

To be determined

Shelf Life

>2 years if stored properly

Drug Formulation

To be determined

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.