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Masupiridine free base

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Specification

Cat. No.

SMD1566

Related Diseases

Schizophrenia

Product Name

Masupiridine free base

Size

Customizable

Price

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Description

Masupiridine, also known as SUVN-502, is a 5-HT6 receptor antagonist under evulation for treating Alzheimer’s disease, attention deficit hyperactivity disorder, Parkinson’s disease and schizophrenia. SUVN-502 is a pure 5-HT6 receptor antagonist with >1200-fold selectivity over 5-HT2A receptor with a superior profile that differentiates from competitor 5-HT6 antagonists. SUVN-502 has an excellent human pharmacokinetics for once a day treatment.

CAS Number

701205-60-9 (free base).

Chemical Formula

C21H24BrN3O3S

Exact Mass

477.0722

Molecular Weight

478.405

Elemental Analysis

C, 52.72; H, 5.06; Br, 16.70; N, 8.78; O, 10.03; S, 6.70

Synonym

SUVN-502; SUVN 502; SUVN502; Masupiridine; Masupiridine free base;

IUPAC/Chemical Name

1-((2-bromophenyl)sulfonyl)-5-methoxy-3-((4-methylpiperazin-1-yl)methyl)-1H-indole

InChi Key

GWCYPEHWIZXYFZ-UHFFFAOYSA-N

InChi Code

InChI=1S/C21H24BrN3O3S/c1-23-9-11-24(12-10-23)14-16-15-25(20-8-7-17(28-2)13-18(16)20)29(26,27)21-6-4-3-5-19(21)22/h3-8,13,15H,9-12,14H2,1-2H3

SMILES Code

CN1CCN(CC2=CN(S(=O)(C3=CC=CC=C3Br)=O)C4=C2C=C(OC)C=C4)CC1

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO, not in water

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.