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LY-2624803

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Specification

Cat. No.

SMD1282

Related Diseases

Insomnia

Product Name

LY-2624803

Size

Customizable

Price

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Description

LY2624803 is a 5-HT2A and histamine H1 receptor antagonist from Eli Lilly as part of its product line-up for therapeutics for the central nervous system. LY2624803 is in phase 2 of clinical trials for the treatment of chronic insomnia. LY2624803 has specific histamine and serotonin receptor antagonism and does not produce other unwanted side effects and it also penetrates into the brain well.

CAS Number

879409-35-5

Chemical Formula

C22H25N3O3

Exact Mass

379.1896

Molecular Weight

379.46

Elemental Analysis

C, 69.64; H, 6.64; N, 11.07; O, 12.65

Synonym

LY-2624803; HY-10275; LY2624803; DB-7;

IUPAC/Chemical Name

1-Piperazinepropanoic acid, 4-dibenz(b,f)(1,4)oxazepin-11-yl-alpha,alpha-dimethyl-

InChi Key

UEFWDVMEDFCHGW-UHFFFAOYSA-N

InChi Code

InChI=1S/C22H25N3O3/c1-22(2,21(26)27)15-24-11-13-25(14-12-24)20-16-7-3-5-9-18(16)28-19-10-6-4-8-17(19)23-20/h3-10H,11-15H2,1-2H3,(H,26,27)

SMILES Code

O=C(O)C(C)(C)CN1CCN(C2=NC3=CC=CC=C3OC4=CC=CC=C24)CC1

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.