Related Diseases
Schizophrenia
Description
Lidanserin is a potential antihypertensive compound which combines vasodilatatory effects due to selective alpha 1-receptor antagonistic action and platelet antiaggregatory, antivasospastic, and vasoprotective properties due to selective 5-HT2-receptor blockade.
Chemical Formula
C26H31FN2O4
Molecular Weight
454.5424
Elemental Analysis
C, 68.70; H, 6.87; F, 4.18; N, 6.16; O, 14.08
Synonym
Lidanserin; ZK 33839; ZK-33839; ZK33839; Lidanserinum; Lidanserine; Lidanserina;
IUPAC/Chemical Name
4-(3-(3-(4-(4-fluorobenzoyl)piperidin-1-yl)propoxy)-4-methoxyphenyl)pyrrolidin-2-one
InChi Key
JDYWZVJXSMADHP-UHFFFAOYSA-N
InChi Code
InChI=1S/C26H31FN2O4/c1-32-23-8-5-20(21-16-25(30)28-17-21)15-24(23)33-14-2-11-29-12-9-19(10-13-29)26(31)18-3-6-22(27)7-4-18/h3-8,15,19,21H,2,9-14,16-17H2,1H3,(H,28,30)
SMILES Code
O=C1NCC(C2=CC=C(OC)C(OCCCN3CCC(C(C4=CC=C(F)C=C4)=O)CC3)=C2)C1
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).
HS Tariff Code
2934.99.9001