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Ketanserin

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Specification

Cat. No.

SMD919

Related Diseases

Depression

Product Name

Ketanserin

Size

100.0mg; 200.0mg; 500.0mg; 1.0g

Price

Inquiry

Availability

2 Weeks

Description

Ketanserin is a 5-HT2A receptor antagonist and potential α1-adrenergic receptor antagonist used to treat hypertension. It decreases blood pressure, improves left ventricular remodeling, increases capillary density in myocardial tissue, and may suppress TRPV1 channel-evoked thermal hyperalgesia.

CAS Number

74050-98-9 (free base)

Chemical Formula

C22H22FN3O3

Exact Mass

395.1645

Molecular Weight

395.43

Elemental Analysis

C, 66.82; H, 5.61; F, 4.80; N, 10.63; O, 12.14

Synonym

Ketanserin; R 41468; R-41468; R41468;

IUPAC/Chemical Name

3-(2-(4-(4-fluorobenzoyl)piperidin-1-yl)ethyl)quinazoline-2,4(1H,3H)-dione

InChi Key

FPCCSQOGAWCVBH-UHFFFAOYSA-N

InChi Code

InChI=1S/C22H22FN3O3/c23-17-7-5-15(6-8-17)20(27)16-9-11-25(12-10-16)13-14-26-21(28)18-3-1-2-4-19(18)24-22(26)29/h1-8,16H,9-14H2,(H,24,29)

SMILES Code

O=C(N1CCN2CCC(C(C3=CC=C(F)C=C3)=O)CC2)NC4=C(C=CC=C4)C1=O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.