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Imagabalin

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Specification

Cat. No.

SMD209

Related Diseases

Anxiety

Product Name

Imagabalin

Size

Customizable

Price

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Description

Imagabalin, also known as PD0332334 and PF-00195889, is a drug which acts as a ligand for the α2δ subunit of the voltage-dependent calcium channel, with some selectivity for the α2δ1 subunit over α2δ2. Imagabalin has demonstrated preclinical efficacy of anxiolytic, analgesic, hypnotic, and anticonvulsant-like activity and is currently in phase III clinical trials for the treatment of generalized anxiety disorder.

CAS Number

610300-07-7

Chemical Formula

C9H19NO2

Exact Mass

173.1416

Molecular Weight

173.256

Elemental Analysis

C, 62.39; H, 11.05; N, 8.08; O, 18.47

Synonym

PD 0332334; PD0332334; PD-0332334; PD 332334; PD332334; PD-332334; PF-00195889; PF 00195889; PF00195889; PF-195889; PF 195889; PF195889; Imagabalin.

IUPAC/Chemical Name

(3S,5R)-3-amino-5-methyloctanoic acid

InChi Key

JXEHXYFSIOYTAH-SFYZADRCSA-N

InChi Code

InChI=1S/C9H19NO2/c1-3-4-7(2)5-8(10)6-9(11)12/h7-8H,3-6,10H2,1-2H3,(H,11,12)/t7-,8+/m1/s1

SMILES Code

CCC[C@@H](C)C[C@H](N)CC(O)=O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO, not in water

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.