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GSK-239512

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Specification

Cat. No.

SMD1544

Related Diseases

Schizophrenia

Product Name

GSK-239512

Size

Customizable

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Description

GSK-239512 is a novel histamine H(3) receptor antagonist. GSK-239512 was developed for the treatment of cognitive dysfunction in neurodegenerative disorders with mild to moderate Alzheimer's disease.

CAS Number

720691-69-0

Chemical Formula

C23H27N3O2

Exact Mass

377.21033

Molecular Weight

377.48

Elemental Analysis

C, 73.18; H, 7.21; N, 11.13; O, 8.48

Synonym

GSK-239512; GSK239512; GSK 239512;

IUPAC/Chemical Name

2-Pyrrolidinone, 1-(6-((3-cyclobutyl-2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)oxy)-3-pyridinyl)-

InChi Key

YFRBKEVUUCQYOW-UHFFFAOYSA-N

InChi Code

InChI=1S/C23H27N3O2/c27-23-5-2-12-26(23)20-7-9-22(24-16-20)28-21-8-6-17-10-13-25(19-3-1-4-19)14-11-18(17)15-21/h6-9,15-16,19H,1-5,10-14H2

SMILES Code

O=C1CCCN1c2ccc(Oc3ccc4CCN(CCc4c3)C5CCC5)nc2

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.