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EVT-101 free base

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Specification

Cat. No.

SMD820

Related Diseases

Depression

Product Name

EVT-101 free base

Size

Customizable

Price

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Description

EVT-101, also known as ENS-101, is an experimental medication which originated from Roche and is under development by Evotec AG for the treatment of major depressive disorder. It acts as a selective NMDA receptor subunit 2B (NR2B) antagonist.

CAS Number

627525-33-1 (free base)

Chemical Formula

C16H13F3N4

Exact Mass

318.1092

Molecular Weight

318.3032

Elemental Analysis

C, 60.38; H, 4.12; F, 17.91; N, 17.60

Synonym

EVT-101 free base; EVT-101; EVT 101; EVT101; ENS-101; ENS 101; ENS101;

IUPAC/Chemical Name

5-(3-Difluoromethyl-4-fluorophenyl)-3-(2-methylimidazol-1-ylmethyl)pyridazine

InChi Key

BOVUHBFXPNLTKF-UHFFFAOYSA-N

InChi Code

InChI=1S/C16H13F3N4/c1-10-20-4-5-23(10)9-13-6-12(8-21-22-13)11-2-3-15(17)14(7-11)16(18)19/h2-8,16H,9H2,1H3

SMILES Code

CC1=NC=CN1CC2=NN=CC(C3=CC=C(F)C(C(F)F)=C3)=C2

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>3 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.