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Enerisant HCl

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Specification

Cat. No.

SMD1509

Related Diseases

Schizophrenia

Product Name

Enerisant HCl

Size

Customizable

Price

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Description

Enerisant HCl is the salt form of Enerisant, a histamine H3 receptor antagonist. In H3 receptor binding assay using (R)-α-methyl[3H]histamine, Enerisant showed IC50 of 4.9 nM. Enerisant may be useful for the treatment of Alzheimer's disease, schizophrenia, etc.

CAS Number

152749-07-9 (HCl)

Chemical Formula

C22H31ClN4O3

Molecular Weight

434.97

Elemental Analysis

C, 60.75; H, 7.18; Cl, 8.15; N, 12.88; O, 11.03

Synonym

Enerisant HCl; Enerisant hydrochloride;

IUPAC/Chemical Name

Methanone, (1-(4-(3-((2R)-2-methyl-1-pyrrolidinyl)propoxy)phenyl)-1H-pyrazol-4-yl)-4-morpholinyl-, hydrochloride (1:1)

InChi Key

QVMTVPSORZKQPZ-GMUIIQOCSA-N

InChi Code

InChI=1S/C22H30N4O3.ClH/c1-18-4-2-9-24(18)10-3-13-29-21-7-5-20(6-8-21)26-17-19(16-23-26)22(27)25-11-14-28-15-12-25;/h5-8,16-18H,2-4,9-15H2,1H3;1H/t18-;/m1./s1

SMILES Code

O=C(C1=CN(C2=CC=C(OCCCN3[C@H](C)CCC3)C=C2)N=C1)N4CCOCC4.[H]Cl

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

To be determined

Shelf Life

>2 years if stored properly

Drug Formulation

To be determined

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.