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Elpetrigine

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Specification

Cat. No.

SMD847

Related Diseases

Depression

Product Name

Elpetrigine

Size

Customizable

Price

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Description

Elpetrigine, also known as GW 273293 and JZP-4, is a potent calcium and sodium channel blocker, which is currently being evaluated in patients as an anticonvulsant and mood stabilizer. JZP-4 could have anxiolytic effects in addition to the anticonvulsant, antidepressant and antimania effects reported earlier.

CAS Number

212778-82-0

Chemical Formula

C10H7Cl3N4

Exact Mass

287.9736

Molecular Weight

289.544

Elemental Analysis

C, 41.48; H, 2.44; Cl, 36.73; N, 19.35

Synonym

GW273293; GW-273293; GW 273293; JZP-4; JZP 4; JZP4; Elpetrigine.

IUPAC/Chemical Name

3-(2,3,5-trichlorophenyl)pyrazine-2,6-diamine

InChi Key

NNXUYJFHOVCRSM-UHFFFAOYSA-N

InChi Code

InChI=1S/C10H7Cl3N4/c11-4-1-5(8(13)6(12)2-4)9-10(15)17-7(14)3-16-9/h1-3H,(H4,14,15,17)

SMILES Code

NC1=NC(N)=CN=C1C2=CC(Cl)=CC(Cl)=C2Cl

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO, not in water

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.