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Devazepide

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Specification

Cat. No.

SMD031

Related Diseases

Anorexia

Product Name

Devazepide

Size

5.0mg; 10.0mg; 25.0mg

Price

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Availability

2 Weeks

Description

Devazepide is a potent, and orally active CCK1 (CCK-A) receptor antagonist that displays appetite-stimulant effects. It blocks the anorectic response to CCK-8 and increases food intake in rats following systemic and i.c.v administration.

CAS Number

103420-77-5

Chemical Formula

C25H20N4O2

Exact Mass

408.15863

Molecular Weight

408.45

Elemental Analysis

C, 73.51; H, 4.94; N, 13.72; O, 7.83

Synonym

Devazepide; Devazepide [USAN:INN]; L 364,718; L 364718; L-364,718; MK 329; MK-329; UNII-JE6P7QY7NH.

IUPAC/Chemical Name

(S)-N-(2,3-Dihydro-1-methyl-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-yl)indole-2-carboxamide

InChi Key

NFHRQQKPEBFUJK-HSZRJFAPSA-N

InChi Code

InChI=1S/C25H20N4O2/c1-29-21-14-8-6-12-18(21)22(16-9-3-2-4-10-16)27-23(25(29)31)28-24(30)20-15-17-11-5-7-13-19(17)26-20/h2-15,23,26H,1H3,(H,28,30)/t23-/m1/s1

SMILES Code

CN1C(=O)[C@@H](NC(=O)c2cc3ccccc3[nH]2)N=C(c4ccccc4)c5ccccc15

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO, not in water

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.