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CP-809101 HCl

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Specification

Cat. No.

SMD553

Related Diseases

Bipolar Disorder

Related Diseases

Depression

Product Name

CP-809101 HCl

Size

10.0mg; 25.0mg; 50.0mg

Price

Inquiry

Availability

2 Weeks

Description

CP-809101 is a potent and selective 5-HT2C receptor agonist (pEC50 values are 9.96, 7.19 and 6.81 for human 5-HT2C, 5-HT2B and 5-HT2A receptors respectively). CP-809101 reduce motor impulsivity and reinstatement of food seeking behavior in male rats. CP-809101 (0.3-3 mg/kg SC) reduced responding for both nicotine and food and blocked the discriminative stimulus properties of nicotine in a similar manner to lorcaserin and Ro 60-0175.

CAS Number

1215721-40-6 (HCl); 479683-64-2 (free).

Chemical Formula

C15H18Cl2N4O

Molecular Weight

341.236

Elemental Analysis

C, 52.80; H, 5.32; Cl, 20.78; N, 16.42; O, 4.69

Synonym

CP-809101; CP 809101; CP809101. CP-809101 HCl; C-809101 HCl; CP 809101 HCl; CP-809101 hydrochloride;

IUPAC/Chemical Name

2-[(3-Chlorophenyl)methoxy]-6-(1-piperazinyl)pyrazine hydrochloride

InChi Key

NMUNRTCTDLORDR-UHFFFAOYSA-N

InChi Code

InChI=1S/C15H17ClN4O.ClH/c16-13-3-1-2-12(8-13)11-21-15-10-18-9-14(19-15)20-6-4-17-5-7-20;/h1-3,8-10,17H,4-7,11H2;1H

SMILES Code

ClC1=CC(COC2=NC(N3CCNCC3)=CN=C2)=CC=C1.[H]Cl

Appearance

Solid powder

Purity

>95% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO, not in water

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.