Related Diseases
Depression
Description
CP-601927 is a nicotinic acetylcholine receptor (nAChR) agonist. It is CNS-penetrant, high affinity, and selective (> 39fold-affinity).
CAS Number
357425-02-6, (free base)
Chemical Formula
C12H12F3N
Elemental Analysis
C, 63.43; H, 5.32; F, 25.08; N, 6.16
Synonym
CP-601927; CP 601927; CP601927; CP-601,927; UNII-VI5LR1EU47.
IUPAC/Chemical Name
(1R,5S)-7-(trifluoromethyl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[d]azepine
InChi Key
RNOBTWYQAWEZHH-JGVFFNPUSA-N
InChi Code
InChI=1S/C12H12F3N/c13-12(14,15)9-1-2-10-7-3-8(6-16-5-7)11(10)4-9/h1-2,4,7-8,16H,3,5-6H2/t7-,8+/m0/s1
SMILES Code
FC(C1=CC=C2[C@](C3)([H])CNC[C@]3([H])C2=C1)(F)F
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO, not in water
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).
HS Tariff Code
2934.99.9001