Inquiry

* Name

Phone

* Email

* Services or Products of Interest

Project Description

* Please note that all of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.

* Tick to confirm the Research Use Only (RUO) statement.

CGP 36742

Inquiry

Specification

Cat. No.

SMD726

Related Diseases

Depression

Product Name

CGP 36742

Size

5.0mg; 10.0mg; 25.0mg

Price

Inquiry

Availability

2 Weeks

Description

CGP36742 is the first orally active GABAB-selective antagonist. CGP 36742's IC50 for blocking GABAergic transmission is 36 μM. CGP36742 in rats blocks baclofen-induced neuronal depression, and reduces learning deficit and passive avoidance in an olfactory bulbectomy depression model.

CAS Number

123690-78-8

Chemical Formula

C7H18NO2P

Exact Mass

179.1075

Molecular Weight

179.2

Elemental Analysis

C, 46.92; H, 10.13; N, 7.82; O, 17.86; P, 17.28

Synonym

CGP 36742; CGP36742; CGP-36742.

IUPAC/Chemical Name

3-aminopropyl-butylphosphinic acid

InChi Key

ONNMDRQRSGKZCN-UHFFFAOYSA-N

InChi Code

InChI=1S/C7H18NO2P/c1-2-3-6-11(9,10)7-4-5-8/h2-8H2,1H3,(H,9,10)

SMILES Code

O=P(CCCC)(CCCN)O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.