XL147 analogue

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Cat. No.: DIA-0230037

Size: 50 mg Size: 500 mg Size: Customer Size

Product Information
CAS No.	956958-53-5
Synonyms	SAR245408
Formula	C₂₁H₁₆N₆O₂S₂
Molecular Weight	448.52
SMILES	CC1=CC=C(C=C1)[S](=O)(=O)NC2=NC3=CC=CC=C3N=C2NC4=CC5=NSN=C5C=C4
Target	PI3Kβ
Product Description	XL147 analogue is a selective and reversible class I PI3K inhibitor for PI3Kα/δ/γ with IC50 of 39 nM/36 nM/23 nM in cell-free assays, less potent to PI3Kβ. Phase 1/2.

Format & Storage
Purity	> 98%
Shipping	Shipped on dry ice.
Storage	Powder: -20 °C, 3 years; 4 °C, 2 years In solvent: -80 °C, 6 months; -20 °C, 1 month
Solubility Overview	Soluble in DMSO

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