WP1066

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Cat. No.: DIA-0230049

Size: 50 mg Size: 500 mg Size: Customer Size

Product Information
CAS No.	857064-38-1
Formula	C₁₇H₁₄BrN₃O
Molecular Weight	356.22
SMILES	CC(NC(=O)\C(=C\C1=NC(=CC=C1)Br)C#N)C2=CC=CC=C2
Target	JAK2 and STAT3
Product Description	WP1066 is a novel inhibitor of JAK2 and STAT3 with IC50 of 2.30 μM and 2.43 μM in HEL cells shows activity to JAK2, STAT3, STAT5, and ERK1/2 not JAK1 and JAK3. Phase 1.

Format & Storage
Purity	> 99%
Shipping	Shipped on dry ice.
Storage	Powder: -20 °C, 3 years; 4 °C, 2 years In solvent: -80 °C, 6 months; -20 °C, 1 month
Solubility Overview	Soluble in DMSO

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