Serabelisib (INK-1117,MLN-1117,TAK-117)

Serabelisib (INK-1117,MLN-1117,TAK-117)

Cat. No.: DIA-0230262

Size: 50 mg Size: 500 mg Size: Customer Size
Product Information
CAS No. 1268454-23-4
Formula C19H17N5O3
Molecular Weight 363.37
SMILES NC1=NC2=C(O1)C=CC(=C2)C3=C[N]4C(=NC=C4C(=O)N5CCOCC5)C=C3
Product Description Serabelisib (INK-1117,MLN-1117,TAK-117) is a potent and selective oral PI3Kα isoform inhibitor (IC50 of 21 nmol/L against PI3Kα) that has demonstrated > 100-fold selectivity relative to other class I PI3K family members (PI3Kβ/γ/δ) and mTOR, and a high degree of selectivity against many other kinase.
Format & Storage
Purity > 98%
Shipping Shipped on dry ice.
Storage Powder: -20 °C, 3 years; 4 °C, 2 years In solvent: -80 °C, 6 months; -20 °C, 1 month
Solubility Overview Soluble in DMSO
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