PIK-75 HCl

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Cat. No.: DIA-0230414

Size: 50 mg Size: 500 mg Size: Customer Size

Product Information
CAS No.	372196-77-5
Formula	C₁₆H₁₅BrClN₅O₄S
Molecular Weight	488.74
SMILES	Cl.CN(/N=C/C1=CN=C2C=CC(=C[N]12)Br)[S](=O)(=O)C3=C(C)C=CC(=C3)[N+]([O-])=O
Product Description	PIK-75 HCl is a p110α inhibitor with IC50 of 5.8 nM (200-fold more potently than p110β), isoform-specific mutants at Ser773, and also potently inhibits DNA-PK with IC50 of 2 nM in cell-free assays.

Format & Storage
Purity	> 98%
Shipping	Shipped on dry ice.
Storage	Powder: -20 °C, 3 years; 4 °C, 2 years In solvent: -80 °C, 6 months; -20 °C, 1 month
Solubility Overview	Soluble in DMSO

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