Pictilisib (GDC-0941)

Inquiry

Cat. No.: DIA-0230417

Size: 50 mg Size: 500 mg Size: Customer Size

Product Information
CAS No.	957054-30-7
Synonyms	RG7321
Formula	C₂₃H₂₇N₇O₃S₂
Molecular Weight	513.64
SMILES	C[S](=O)(=O)N1CCN(CC1)CC2=CC3=NC(=NC(=C3S2)N4CCOCC4)C5=CC=CC6=C5C=N[NH]6
Target	PI3Kα/δ
Product Description	Pictilisib (GDC-0941) is a potent inhibitor of PI3Kα/δ with IC50 of 3 nM in cell-free assays, with modest selectivity against p110β (11-fold) and p110γ (25-fold). Phase 2.

Format & Storage
Purity	> 98%
Shipping	Shipped on dry ice.
Storage	Powder: -20 °C, 3 years; 4 °C, 2 years In solvent: -80 °C, 6 months; -20 °C, 1 month
Solubility Overview	Soluble in DMSO

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.