PDHK-IN-5

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Cat. No.: DIA-0243309

Size: 50 mg Size: 100 mg Size: 250 mg Size: Customer Size

Product Information
Formula	C₃₀H₃₁N₅O₂
Molecular Weight	493.60
SMILES	CC1=NC2=C(C3=CC=CC(C4CC4)=C3N2)C=C1C5=NN=C(O5)C(C(C)C)CC(NCC6=CC=CC=C6)=O
Target	PDHK
Product Description	PDHK-IN-5 (Compound 19) is a potent inhibitor of PDHK with IC50s of 0.006 and 0.0329 μM for PDHK2 and PDHK4, repectively. Pyruvate dehydrogenase kinases (PDHKs) are fascinating agent targets for numerous diseases, including diabetes and cancers. PDHK-IN-5 has the potential for the research of cancer diseases.

Format & Storage
Shipping	Room temperature in the continental U.S. Other areas may vary.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.