GSK2656157

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Cat. No.: DIA-0230792

Size: 50 mg Size: 500 mg Size: Customer Size

Product Information
CAS No.	1337532-29-2
Formula	C₂₃H₂₁FN₆O
Molecular Weight	416.45
SMILES	C[N]1C=C(C2=C(F)C3=C(C=C2)N(CC3)C(=O)CC4=CC=CC(=N4)C)C5=C(N)N=CN=C15
Product Description	GSK2656157 is an ATP-competitive and highly selective inhibitor of PERK with IC50 of 0.9 nM in a cell-free assay, 500-fold greater against a panel of 300 kinases.

Format & Storage
Purity	> 98%
Shipping	Shipped on dry ice.
Storage	Powder: -20 °C, 3 years; 4 °C, 2 years In solvent: -80 °C, 6 months; -20 °C, 1 month
Solubility Overview	Soluble in DMSO

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