GRK5-IN-3

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Cat. No.: DIA-0230802

Size: 100 mg Size: 500 mg Size: Customer Size

Product Information
CAS No.	2410793-22-3
Formula	C₂₃H₂₁N₇O₃
Molecular Weight	443.46
Target	GRK5 and GRK6
Product Description	GRK5-IN-3 is a covalent inhibitor of GRK5 (G Protein-Coupled Receptor Kinase 5). GRK5-IN-3 shows potent inhibitory effect to GRK5 and GRK6 with IC50s of 0.22 μM and 0.41 μM, respectively.

Format & Storage
Format	Solid
Purity	> 99%
Shipping	Shipped on dry ice.
Storage	Protect from light. Powder: -80 °C, 2 years; -20 °C, 1 year. In solvent: -80 °C, 6 months; -20 °C, 1 month (protect from light).
Solubility Overview	Soluble in DMSO

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