Cat. No.: DIA-0243087
Product Information | |
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CAS No. | 332117-28-9 |
Synonyms | TCS 5861528 |
Formula | C19H23N5O3 |
Molecular Weight | 369.42 |
SMILES | O=C1C2=C(N=CN2CC(NC3=CC=C(C(C)CC)C=C3)=O)N(C)C(N1C)=O |
Target | TRP Channel |
Product Description | Chembridge-5861528 (TCS 5861528) is a potent TRPA1 channel antagonist that antagonizes similarly allyl isothiocyanate- and 4-HNE-evoked TRPA1 responses, with IC50 values of 14.3 μM and 18.7 μM, respectively. Chembridge-5861528 shows antihypersensitivity activities. |
Format & Storage | |
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Format | Solid |
Color | White to off-white |
Purity | 99.76% |
Shipping | Room temperature in the continental U.S. Other areas may vary. |
Storage | Powder: -20°C, 3 years; 4°C, 2 years In solvent: -80°C, 2 years; -20°C, 1 year |
Solubility Overview | Soluble in DMSO |
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