Cat. No.: DIA-0231339
Product Information | |
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CAS No. | 870281-34-8 |
Synonyms | CAL-120 |
Formula | C21H16FN7O |
Molecular Weight | 401.4 |
SMILES | CC(NC1=NC=NC2=C1[NH]C=N2)C3=NC4=C(C=C(F)C=C4)C(=O)N3C5=CC=CC=C5 |
Target | p110δ |
Product Description | acalisib (GS-9820) is a highly selective and potent p110δ inhibitor (IC50 = 14 nM) with 114- to 400-fold selectivity over the other class I PI3K enzymes and no activity against Class II and III PI3K family members or other PI3K-related proteins including mTOR and DNA-PK. |
Format & Storage | |
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Purity | > 99% |
Shipping | Shipped on dry ice. |
Storage | Powder: -20 °C, 3 years; 4 °C, 2 years In solvent: -80 °C, 6 months; -20 °C, 1 month |
Solubility Overview | Soluble in DMSO |