Rilmenidine hemifumarate
Cat. No: CDIA-0644
CAS. No.: 207572-68-7
Size: 5 mg
| Product Details |
| Formula |
C10H16N2O.1/2C4H4O4 |
| Molecular Weight |
238.28 |
| Appearance |
Solid |
| Purity |
99.78% |
| Smiles String |
O=C(O)/C=C/C(O)=O.C1(NC(C2CC2)C3CC3)=NCCO1.[0.5] |
| Storage & Handling |
| Shipping |
Room temperature. |
| Storage |
-20 °C, stored under nitrogen, away from moisture
*In solvent : -80 °C, 6 months; -20 °C, 1 month (stored under nitrogen, away from moisture) |
Description
Rilmenidine hemifumarate, an innovative antihypertensive agent, is an orally active, selective I1 imidazoline receptor agonist. Rilmenidine hemifumarate is an alpha 2-adrenoceptor agonist. Rilmenidine hemifumarate induces autophagy. Rilmenidine hemifumarate acts both centrally by reducing sympathetic overactivity and in the kidney by inhibiting the Na+/H+ antiport. Rilmenidine hemifumarate modulates proliferation and stimulates the proapoptotic protein Bax thus inducing the perturbation of the mitochondrial pathway and apoptosis in human leukemic K562 cells .
! For research use only. Not intended for any clinical use.
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