Palosuran hydrochloride

Cat. No: CDIA-1721

CAS. No.: 2469274-58-4

Synonyms: ACT-058362 hydrochloride

Size: 50 mg

Price: Inquiry

Product Details
Formula	C25H31ClN4O2
Molecular Weight	454.99
Appearance	Solid
Purity	98.67%
Smiles String	OC(CC1=CC=CC=C1)(CC2)CCN2CCNC(NC3=CC(C)=NC4=CC=CC=C34)=O.[H]Cl

Storage & Handling
Shipping	Room temperature.
Storage	4 °C, sealed storage, away from moisture *In solvent : -80 °C, 6 months; -20 °C, 1 month (sealed storage, away from moisture)

Description

Palosuran hydrochloride (ACT-058362 hydrochloride) is a potent, selective, and orally active antagonist of urotensin II receptor, with an IC50 of 3.6 nM for CHO cell membranes expressing human recombinant receptors. Palosuran hydrochloride can improves pancreatic and renal function in diabetic rats.

! For research use only. Not intended for any clinical use.