MRS2179 tetrasodium hydrate

Product Details
Formula	C11H13N5O9P2Na4.3?H2O
Molecular Weight	576.21
Appearance	Solid
Purity	≥99.0%
Smiles String	CNC1=C2C(N([[email protected]](C[[email protected]@H]3O[P](O[Na])(O[Na])=O)([H])O[[email protected]@H]3CO[P](O[Na])(O[Na])=O)C=N2)=NC=N1.O.[3.5]

Storage & Handling
Shipping	Room temperature.
Storage	-20 °C, sealed storage, away from moisture *In solvent : -80 °C, 6 months; -20 °C, 1 month (sealed storage, away from moisture)

MRS2179 tetrasodium hydrate is a competitive P2Y1 receptor antagonist, with a Kb of 102 nM and a pA2 of 6.99 for turkey P2Y1 receptor. MRS2179 tetrasodium hydrate is selective for P2Y1 over P2X1 (IC50=1.15 µM), P2X3 (12.9 µM), P2X2, P2X4, P2Y2, P2Y4, and P2Y6 receptors. MRS2179 tetrasodium hydrate inhibits platelet aggregation.

! For research use only. Not intended for any clinical use.