MRS 1523

Cat. No: CDIA-0742

CAS. No.: 212329-37-8

Size: 5 mg

Price: Inquiry

Product Details
Formula	C23H29NO3S
Molecular Weight	399.55
Appearance	Oil
Purity	99.93%
Smiles String	O=C(OCCC)C1=C(C(C(SCC)=O)=C(N=C1C2=CC=CC=C2)CC)CCC

Storage & Handling
Shipping	Room temperature.
Storage Pure Form	-20 °C/3 years\|\|\|\|4 °C/2 years

Description

MRS 1523 is a potent and selective adenosine A3 receptor antagonist with Ki values of 18.9 nM and 113 nM for human and rat A3 receptors, respectively. In rat this corresponds to selectivities of 140- and 18-fold vs A1 and A2A receptors, respectively. MRS 1523 can exert antihyperalgesic effect through N-type Ca channel block and action potential inhibition in isolated rat dorsal root ganglion (DRG) neurons.

! For research use only. Not intended for any clinical use.