GSK5182

Cat. No: CDIA-0697

CAS. No.: 877387-37-6

Size: 5 mg

Price: Inquiry

Product Details
Formula	C27H31NO3
Molecular Weight	417.54
Appearance	Solid
Purity	99.85%
Smiles String	OCCC/C(C1=CC=CC=C1)=C(C2=CC=C(O)C=C2)/C3=CC=C(OCCN(C)C)C=C3.[(Z)]

Storage & Handling
Shipping	Room temperature.
Storage Powder	-20 °C/3 years, 4 °C/2 years

Description

GSK5182 is a highly selective and orally active inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM. GSK5182 does not interact with other nuclear receptors, including ERRα or ERα. GSK5182 also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma (HCC).

! For research use only. Not intended for any clinical use.