GRK5-IN-4
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GRK5-IN-4

Cat. No: CDIA-1954
CAS. No.: 2410794-89-5
Synonyms: CCG-265328
Size: 50 mg
Price: Inquiry
Product Details
Formula C26H25N7O3
Molecular Weight 483.52
Smiles String O=C(NCC1=CC=C(C(OC)=C1)NC2=NC(NC3=C(C(NC)=O)C=CC=C3)=C4C=CNC4=N2)C#CC
Storage & Handling
Shipping Room temperature.
Storage Please refer to the instruction manual.

Description

GRK5-IN-4 (Compound 16d, CCG-265328) is a potent and and selective covalent GRK5 (G protein-coupled receptor kinase 5) inhibitor, with an IC50 of 1.1 μM. GRK5-IN-4 shows 90-fold selectivity over GRK2. GRK5-IN-4 can be used for heart failure research.

! For research use only. Not intended for any clinical use.