(E/Z)-GSK5182

Cat. No: CDIA-0800

Size: 100 mg

Price: Inquiry

Product Details
Formula	C27H31NO3
Molecular Weight	417.54
Appearance	Solid
Purity	99.17%
Smiles String	OCCC/C(C1=CC=CC=C1)=C(C2=CC=C(C=C2)OCCN(C)C)\C3=CC=C(C=C3)O

Storage & Handling
Shipping	Room temperature.
Storage Powder	-20 °C/3 years, 4 °C/2 years

Description

(E/Z)-GSK5182 is a racemic compound of (E)-GSK5182 and (Z)-GSK5182 isomers. GSK5182 is a highly selective and orally active inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM. GSK5182 also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma.

! For research use only. Not intended for any clinical use.