Enoximone
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Enoximone

Cat. No: CDIA-0667
CAS. No.: 77671-31-9
Size: 100 mg
Price: Inquiry
Product Details
Formula C12H12N2O2S
Molecular Weight 248.30
Appearance Solid
Purity 98.05%
Smiles String O=C1NC(C)=C(C(C2=CC=C(SC)C=C2)=O)N1
Storage & Handling
Shipping Room temperature.
Storage Powder -20 °C/3 years, 4 °C/2 years

Description

Enoximone is an inotropic vasodilating agent and a selective and orally active phosphodiesterase III (PDE3) inhibitor with an IC50 of 5.9 μM. Enoximone induces vasodilatation and increases intracellular levels of cAMP by inhibiting cGMP-inhibited PDE. Enoximone also exhibits PDE4 inhibitory effect with an IC50 of 21.1 μM for myocardial PDE4A. Enoximone has the potential for congestive heart failure research and has bronchodilatory, antiasthma and anti-inflammatory effects.

! For research use only. Not intended for any clinical use.