CMPD101

Cat. No: CDIA-0438

CAS. No.: 865608-11-3

Size: 10 μg

Price: Inquiry

Product Details
Formula	C24H21F3N6O
Molecular Weight	466.46
Appearance	Solid
Purity	98.74%
Smiles String	O=C(C1=CC(NCC2=NN=C(C3=CC=NC=C3)N2C)=CC=C1)NCC4=CC=CC=C4C(F)(F)F

Storage & Handling
Shipping	Room temperature.
Storage Powder	-20 °C/3 years, 4 °C/2 years

Description

CMPD101 is a potent, highly selective and membrane-permeable small-molecule inhibitor of GRK2/3 with IC50 of 18 nM and 5.4 nM, respectively. CMPD101 exhibits less selectively against GRK1, GRK5, ROCK-2 and PKCα with IC50s of 3.1 μM , 2.3 μM, 1.4 μM and 8.1 μM, respectively. CMPD101 can be used for the study of heart failure.

! For research use only. Not intended for any clinical use.