Azepexole di hydrochloride
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Azepexole di hydrochloride

Cat. No: CDIA-1693
CAS. No.: 36067-72-8
Synonyms: B-HT 933 dihydrochloride; Oxazoloazepin dihydrochloride
Size: 50 mg
Price: Inquiry
Product Details
Formula C9H17Cl2N3O
Molecular Weight 254.16
Smiles String NC(O1)=NC2=C1CCN(CC)CC2.[H]Cl.[H]Cl
Storage & Handling
Shipping Room temperature.
Storage Please refer to the instruction manual.

Description

Azepexole (B-HT 933) dihydrochloride is a potent and selective alpha 2-adrenoceptor agonist with pKis of 8.3, 7.6, and 7.5 for α2A-, α2B- and α2C-adrenoceptor subtypes, resepctively. Azepexole dihydrochloride causes concentration-dependent inhibition of peristaltic contractions (IC50= 78.72 nM).

! For research use only. Not intended for any clinical use.