ARC 239 di hydrochloride
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ARC 239 di hydrochloride

Cat. No: CDIA-1855
CAS. No.: 55974-42-0
Size: 50 mg
Price: Inquiry
Product Details
Formula C24H31Cl2N3O3
Molecular Weight 480.43
Appearance Solid
Purity 99.57%
Smiles String O=C1C2=C(C(C)(C)C(N1CCN3CCN(CC3)C4=C(OC)C=CC=C4)=O)C=CC=C2.Cl.Cl
Storage & Handling
Shipping Room temperature.
Storage 4 °C, sealed storage, away from moisture *In solvent : -80 °C, 6 months; -20 °C, 1 month (sealed storage, away from moisture)

Description

ARC 239 dihydrochloride is a selective α2B/2C adrenoceptor antagonist (pKd values are 5.95, 7.41 and 7.56 at α2A, α2B, and α2C receptors respectively). ARC 239 dihydrochloride binds to CHO cell membranes expressing human recombinant a2A-, a2B- or a2C-adrenoceptor subtypes with pKis of 5.6, 8.4, and 7.08, respectively.

! For research use only. Not intended for any clinical use.